Found 88 of ec50 data for polymerid = 49000904 TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.0200nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.0600nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.0600nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.0700nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.0800nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.120nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at PTH1 receptor (unknown origin) assessed as induction of cAMPMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.140nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.150nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.150nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.180nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl-cyclase activity after 4...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.260nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.290nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.300nMAssay Description:Agonist activity at PTH1R overexpressed in HEK293 cells assessed as intracellular cAMP productionMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.320nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.340nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.360nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.440nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.480nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.510nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.510nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.520nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.650nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.710nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.790nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.830nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 0.920nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at PTH1R overexpressed in HEK293 cells assessed as intracellular cAMP mobilizationMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in HEK293 cells assessed as induction of luciferase activity by CRE-luciferase reporter ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 2.20nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl-cyclase activity after 4...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Agonist activity at recombinant human PTHR1 expressed in pig LLC-PK1 cells assessed as increase in cAMP production measured after 20 mins by EIAMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 2.5nMAssay Description:Agonist activity at human PTHR1 expressed in HKRKB7 cells assessed as accumulation of intracellular cAMP after 20 mins by enzyme immunoassayMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 2.60nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 4.40nMAssay Description:Partial agonist activity at human PTH receptor expressed in OK-1 cells assessed as increase in cAMP productionMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at human PTH1 receptor expressed in human GP2.3 cells assessed as induction of cAMP after 12 to 20 mins by luciferase reporter gene ...More data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 5.5nMAssay Description:Partial agonist activity at human PTH receptor expressed in OK-1 cells assessed as increase in cAMP productionMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 7.20nMAssay Description:Activity at human PTH/PTH-related peptide receptor expressed in SAOS2 cells assessed as cAMP formationMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University of Wisconsin-Madison
Curated by ChEMBL
University of Wisconsin-Madison
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Partial agonist activity at human PTH receptor expressed in OK-1 cells assessed as increase in cAMP productionMore data for this Ligand-Target Pair
